Publikációk 2015

   1. Tímea Magyar, Ferenc Miklós, László Lázár, Ferenc Fülöp:
       Application of a ball milling technique for the condensation of anthranilic hydrazides with aromatic aldehydes towards 4-quinazolinone derivatives
      Chem. Heterocycl. Comp., 50, 1463-1469 (2015)
   2. István Ilisz, Nóra Grecsó, Aleksandra Misicka, Dagmara Tymecka, László Lázár, Wolfgang Lindner, Antal Péter:
       Comparison of the separation performances of Chinchona alkaloid-based zwitterionic stationary phases in the enantioseparation of β2- and β3
       amino acids

       Molecules, 20, 70-87 (2015)
   3. Elena Stanoeva, Angelina Georgieva, Stanislava Avramova, Nikola Burdzhiev, László Lázár:
       Synthesis of novel 13a-(ɷ-aminoalkyl)-8-oxoberbines by means of reaction of homophthalic anhydride with 1-substituted 3,4
       dihydroisoquinolines. An unexpected formation of a pyrrolo[3,4-

       J. Heterocyclic Chem.,52, 130-135 (2015)
   4. István Baczkó, István Leprán, Loránd Kiss, Danina M. Muntean, Peter E. Light:
       Future perspectives in the pharmacological treatment of atrial fibrillation and venticular arrhythmias in hearth failure
      Curr. Pharm. Design., 21, 1011-1029 (2015)
   5. Danina M. Muntean, Loránd Kiss, Norbert Jost, István Baczkó:
       ATP-sensitive potassium channel modulators and cardiac arrhythmias: an update
      Curr. Pharm. Design., 21, 1091-1102 (2015)
   6. Melinda Nonn, Loránd Kiss, Mikko M. Hänninen, Ferenc Fülöp:
       An insight into the synthesis of novel aryl-substituted alicyclic β-amino acid derivatives through substrate-directed palladium-catalysed regio- and
       stereoselective cross-coupling

      RSC Adv.,5, 13628-13634 (2015)
   7. István Ilisz, Nóra Grecsó, Ferenc Fülöp, Wolfgang Lindner, Antal Péter:
       High-performance liquid chromatographic enantioseparation of cationic 1,2,3,4-tetrahydroisoquinoline analogs on Cinchona alakloid-based
       zwitterionic chiral stationary phases

       Anal. Bioanal. Chem., 407, 961-972 (2015)
   8. Loránd Kiss, Márton Kardos, Enikő Forró, Ferenc Fülöp:
       Stereocontrolled one-step synthesis of difunctionalised cispentacin derivatives through ring-opening metathesis of norbornene β-amino acids
      Eur. J. Org. Chem.,2015, 1283-1289 (2015)
   9. Shan-Han Huang, Chun-Wei Tung, Ferenc Fülöp, Jih-Heng Li:
       Developing a QSAR model for hepatotoxicity screening of the active compounds in traditional Chinese medicines
       Food and Chemical Toxicology, 78, 71-77 (2015)
  10. István Ilisz, Zsanett Gecse, Gyula Lajkó, Melinda Nonn, Ferenc Fülöp, Wolfgang Lindner, Antal Péter:
        Investigation of the structure-selectivity relationships and van’t Hoff analysis of chromatographic stereoisomer separations of unusual isoxazoline
        fused 2-amino­cyclopentanecarboxylic acids on Chinchona alkaloid-based chiral stationary phases

       J. Chromatography A, 1384, 67-75 (2015)
  11. Anita Aranyi, István Ilisz, Antal Péter, Ferenc Fülöp, Caroline West:
        Exploring the enantioseparation of amino-naphthol analogues by supercritical fluid chromatography
        J. Chromatography A 1387, 123-133 (2015)
  12. Melinda Nonn, Loránd Kiss, Matti Haukka, Santos Fustero, Ferenc Fülöp:
        A novel and selective fluoride opening of aziridines by XtalFluor-E. Synthesis of fluorinated diamono acid derivatives
       Org. Lett. 17, 1074-1077 (2015)
  13. Loránd Kiss, Maria Cherepanova, Ferenc Fülöp:
        Recent advances in the stereoselective syntheses of acyclic disubstituted β2,3-amino acids
       Tetrahedron 71, 2049-2069 (2015)
  14. Gábor Olajos, Anasztázia Hetényi, Edit Wéber, Lukács J. Németh, Zsolt Szakonyi, Ferenc Fülöp, Tamás A. Martinek:
        Induced folding of protein-sized foldameric β-sandwich models with core β-amino acid residues
        Chem. Eur J.21, 6173-6180 (2015)
  15. Enikő Forró, Zsolt Galla, Zala Nádasdi, Judit Árva, Ferenc Fülöp:
       Novel chemo-enzymatic route to a key intermediate for the taxol side-chain through enantioselective O-acylation. Unexpected acyl migration
       J. Mol. Cat. B: Enzymatic116, 101-105 (2015)
  16. Nóra Grecsó, István Ilisz, Zsanett Gecse, László Schönstein, Ferenc Fülöp, Antal Péter:
       High-performance liquid chromatographic enantioseparation of amino alcohol analogues possessing 1,2,3,4-tetrahydroisoquinoline skeleton on
       polysaccharide-based chiral stationary phases

       Biomed. Chromatogr. 29, 788-796 (2015)
  17. Zsuzsanna Bohár, József Toldi, Ferenc Fülöp, László Vécsei:
       Changing the face of kynurenines and neurotoxicity: therapeutic considerations
       Int. J. Mol. Sci. 16, 9772-9793 (2015)
  18. Loránd Kiss, Enikő Forró, Ferenc Fülöp:
       Novel stereocontrolled syntheses of tashiromine and epitashiromine
       Beilstein J. Org. Chem. 11, 596-603 (2015)
  19. Krisztina Dobi, Beáta Flachner, Mária Pukáncsik, Enikő Máthé, Melinda Bognár, Mária Szaszkó, Csaba Magyar, István Hajdú, Zsolt Lőrincz, István
Ferenc Fülöp, Sándor Cseh, György Dormán:
       Combination of pharmacophore matching, 2D similarity search and in vitro biological assay in the selection of potential 5-HT6 anatagonists from
       large commercial repositories
       Chem. Biol. Drug. Des. 2015, 1-17 (2015)
  20. Chi-Ting Hsieh, Sándor B. Ötvös, Yang-Chang Wu, István M. Mándity, Fang-Rong Chao, Ferenc Fülöp:
       Highly selective continuous-flow synthesis of potentially bioactive deuterated chalcone derivatives
      ChemPlusChem, 80, 859-864 (2015)
  21. Sándor B. Ötvös, Ádám Georgiádes, Mónika Ádok-Sipiczki, Rebeka Mészáros, István Pálinkó, Pál Sipos, Ferenc Fülöp:
       A layered double hydroxide, a synthetically useful heterogeneous catalyst for azide–alkyne cycloadditions in a continuous-flow reactor
       Applied Catalysis A: General 501, 63-73 (2015)
  22. Zsolt Szakonyi, Árpád Csőr, Matti Haukka, Ferenc Fülöp:
        Stereoselective synthesis of carane-based chiral β- and γ-amino acid derivatives via conjugate addition
       Tetrahedron 71, 4846-4852 (2015)
  23. István Ilisz, Nóra Grecsó, Enikő Forró, Ferenc Fülöp, Daniel W. Armstrong, Antal Péter:
       High-performance liquid chromatographic separation of paclitaxel intermediate phenylisoserine derivatives on macrocyclic glycopeptide and
       cyclofructan-based chiral stationary phases
       J. Pharmaceutical and Biomedical Analysis 114, 312-320 (2015)
  24. Alexandra Petrus, Oana M. Duicu, Adrian Sturza, Lavinia Noveanu, Loránd Kiss, Maria Danila, István Baczkó, Danina M. Muntean, Norbert Jost:
       Modulation of mitochondrial respiratory function and ROS production by novel benzopyran analogues
       Can. J. Physiol. Pharmacol93, 811-818 (2015)
  25. Judit Sas, István Szatmári, Ferenc Fülöp:
       Selective N-alkylation of isoquinolines, benzazepines and thienopyridines with aromatic aldehydes and naphthols
       Tetrahedron 71, 7216-7221 (2015)
  26. Eszter Sélley, Gergő A. Molnár, Szilárd Kun, István András Szijártó, Boglárka Laczy, Tibor Kovács, Ferenc Fülöp, István Wittmann
       Complex vasoactivity of liraglutide. Contribution of three gasotransmitters
       Artery Research 11, 1-9 (2015)
  27. István Ilisz, Zsanett Gecse, Gyula Lajkó, Enikő Forró, Ferenc Fülöp, Wolfgang Lindner, Antal Péter:
       High-performance liquid chromatographic enantioseparation of cyclic β-amino acids on zwitterionic chiral stationary phases based
       in Chinchona alkaloids
       Chirality 27, 563-570 (2015).
  28. Yolanda C. Rodrigez, Tayla M. Duarte, Zsolt Szakonyi, Enikő Forró, Ferenc Fülöp, Thomas J. Wenzel:
       Utilization of (18-crown-6)-2,3,11,12-tetracarboxylic acid as a chiral NMR solvating agent for diamines and β-amino acids
      Chirality 27, 708-715 (2015)
  29. Gyula Lajkó, István Ilisz, Gábor Tóth, Ferenc Fülöp, Wolfgang Lindner, Antal Péter:
        Application of Chinchona alkaloid-based zwitterionic chiral stationary phases in supercritical fluid chromatography for the enantioseparation of Nα
        protected proteinogenic amino acids
        J. Chromatography A 1415, 134-135 (2015)
  30. Krisztina Dobi, Beáta Flachner, Mária Pukáncsik, Enikő Máthé, Melinda Bognár, Mária Szaszkó, Csaba Magyar, István Hajdú, Zsolt Lőrincz, István
       Simon, Ferenc Fülöp, Sándor Cseh, György Dormán:
       Combination of Pharmacophore matching, 2D similarly search, and in vitro biological assays in the selection of potential 5-HT6 antagonists from
       large commercial repositories
       Chem. Biol. Drug Des.86, 864-880 (2015)
  31. Sándor B. Ötvös, Ferenc Fülöp:
       Flow chemistry as a versatile tool for the synthesis of triazoles:
      Catal. Sci. Technol5, 4926-4941 (2015)
  32. Ferenc Miklós, Alexandra Petrisor, Ferenc Fülöp:
        Alternative conditions for the synthesis of novel spiro[1,3-N,N-heterocyclic-adamantanes]
        Arkivoc 158-171 (2015)
  33. Ferenc Kassai, Rita Kedves, István Gyertyán, Bernadett Tuka, Ferenc Fülöp, József Toldi, Balázs Lendvai, László Vécsei:
        Effect of a kynurenic acid analog on home-cage activity and body temperature in rats
       Pharmacological Reports 67, 1188-1192 (2015)
  34. István Mándity, Ferenc Fülöp:
       An overview of peptide and peptoid foldamers in medicinal chemistry
      Expert Opin.Drug Discov10, 1163-1177 (2015)
  35. Sándor B. Ötvös, Alíz Szloszár, István M. Mándity, Ferenc Fülöp:
       Heterogeneous dipeptide-catalyzed α-amination of aldehydes in a continuous-flow reactor: effect of residence time on enantioselectivity
       Adv. Synth. Catal357, 3671-3680 (2015)
  36. Loránd Kiss, Enikő Forró, György Orsy, Renáta Ábrahámi, Ferenc Fülöp:
       Stereo- and regiocontrolled syntheses of exomethylenic cyclohexane β-amino acid derivatives
       Molecules 20, 21094-21102 (2015)
  37. Márton Kardos, Loránd Kiss, Ferenc Fülöp:
       Stereocontrolled synthesis of difunctionalized azetidinones and β2,3-amino acid derivatives from cyclodienes by ring-opening and cross-metathesis
       Asian J. Org. Chem4, 1155-1159 (2015)
  38. Zsolt Fekete, Zsuzsanna Rajnai, Tünde Nagy, Katalin Tauberné Jakab, Anita Kurunczi, Katalin Gémes, Krisztina Herédi-Szabó, Ferenc Fülöp, Gábor
       K. Tóth, Maciej Czerwinski, Greg Loewen, Peter Krajcsi:
       Membrane assays to characterize interaction of drugs withABCB1
       J. Membrane Biol. 248, 967-977 (2015)
  39. A. Csáti, L. Edvinsson, László Vécsei, József Toldi, Ferenc Fülöp, J. Tajti, K. Warfvinge:
       Kynurenic acid modulates experimentally induced inflammation in the trigeminal ganglion
      The Journal of Headache and Pain 1-14 (2015)                                                           
  40. István Ilisz, Nóra Grecsó, Roman Popoušek, Zoltán Pataj, Petr Barták, László Lázár, Ferenc Fülöp, Wolfgang Lindner, Antal Péter:
       High-performance liquid chromatographic separation of unusual β3-amino acid enantiomers in different chromatographic modes
       on Cinchona alkaloid-based zwitterionic chiral stationary phases
      Amino Acids 47, 2279-2291 (2015)                                                                               
  41. Lenke Kovács, György Szőllősi, Ferenc Fülöp:
       Pt–Cinchonidine catalyzed asymmetric catalytic cascade reaction of 2-nitrophenylpyruvates in flow system
      J. Flow. Chem5, 210-215 (2015)