Publikációk 2016

  • Nyomtatás

   1. Zsolt Galla, Ferenc Beke, Enikő Forró, Ferenc Fülöp:
       Enantioselective hydrolysis of 3,4-disubstituted β-lactams. An efficient enzymatic method for the preparation of a key Taxol side-chain intermediate
       J. Mol. Catalysis B: Enzymatic123, 107-112 (2016)
   2. Jurgen Caroen, An Clemmen, Judit Kámán, Fréderique Backaert, Jan L. Goeman, Ferenc Fülöp, Johan Van der Eycken:
       Solid-phase synthesis of 6,7-cycloalkane-fused 1,4-diazepane-2,5-diones via a cyclization/release strategy
       Tetrahedron72, 148-160 (2016)
   3. Szakonyi Zsolt:
       Monoterpénvázas 3-amino-1,2-diolok sztereoszelektív előállítása, átalakításai és alkalmazásai
       Magyar Kémikusok Lapja71, 3-4 (2016)                                                                      
   4. Loránd Kiss, Attila Márió Remete, Melinda Nonn, Santos Fustero, Reijo Sillanpää, Ferenc Fülöp:
       Substrate-dependent fluorinations of highly functionalized cycloalkanes
      Tetrahedron, 72, 781-787 (2016)
   5. Ferenc Miklós, Ferenc Fülöp:
       A simple green protocol for the condensation of anthranilic hydrazide with cyclohexanone and N-benzylpiperidinone in water 
       J. Heterocyclic Chem. 53, 32-37 (2016)
   6. Nóra Grecsó, Michal Kohout, Andrea Carotti, Roccaldo Sardella, Benedetto Natalini, Ferenc Fülöp, Wolfgang Lindner, Antal Péter, István Ilisz:
       Mechanistic considerations of enantiorecognition on novel Cinchona alkaloidbased zwitterionic chiral stationary phases from the aspect of the
       separation of trans-paroxetine enantiomers as model compounds

       J. Pharmaceutical Biomedical Analysis 124, 164-173 (2016)
   7. Sándor B. Ötvös, Chi-Ting Hsieh, Yang-Chang Wu, Jih-Heng Li, Fang-Rong Chang, Ferenc Fülöp:
      Continuous-flow synthesis of deuterium-labeled antidiabetic chalcones: studies towards the selective deuteration of the alkynone core
      Molecules 21, 318-328 (2016)
   8. Petra Barta, István Szatmári, Ferenc Fülöp, Matthias Heydenreich, Andreas Koch, Erich Kleinpeter:
       Synthesis and stereochemistry of new naphth[1,3]oxazino[3,2-a]benzazepine and naphth[1,3]oxazino[3,2-e]thienopyridine derivatives
      Tetrahedron, 72, 2402-2410 (2016)
   9. Gyula Lajkó, Tímea Orosz, Nóra Grecsó, Beáta fekete, Márta Palkó, Ferenc Fülöp, Wolfgang Lindner, Antal Péter, István Ilisz:
       High performance liquid chromatographic enantioseparation of cyclic β-aminohydroxamic acids on zwitterionic chiral stationary phasese based on
       Chinchona alakaloids

       Analytica Chimica Acta 921, 84-94 (2016)
  10. Zsolt Szakonyi, Árpád Csőr, Antal Csámpai, Ferenc Fülöp:
       Stereoselective synthesis and modelling-driven optiomisation of Carane-based aminodiols and 1,3-oxazines as catalysts for the enantioselective
       addition of diethylzinc to benzaldehyde

       Chem. Eur. J.22, 7163-7173 (2016)
  11. Tímea Gonda, Zsolt Szakonyi, Antal Csámpai, Matti Haukka, Ferenc Fülöp:
        Stereoselective synthesis and application of tridentate aminodiols derived from
        (+)-pulegone

        Tetrahedron: Assymetry 27, 480-486 (2016)
  12. Enikő Forró, Zsolt Galla, Ferenc Fülöp:
       The N-hydroxymethyl group as a traceless activating group for the CAL-B-catalysed ring cleavage of β-lactams: atype of two-step cascade reaction
       Eur. J. Org. Chem, 2647-2652 (2016)
  13. Zsófia Hegedűs, Ildikó Makra, Norbert Imre, Anasztázia Hetényi, István M. Mándity, Éva Monostori, Tamás A. Martinek:
       Foldameric probes for membrane interactions by induced β-sheet folding
       Chem. Commun. 52, 1891-1894 (2016)
  14. István M. Mándity, Sándor B. Ötvös, György Szőlősi, Ferenc Fülöp:
        Harnessing the versatility of continuous-flow processes: selective and efficient reactions
       Chem. Rec. 16, 1018-1033 (2016)
  15. Ötvös Sándor Balázs:
        Áramlásos módszerekkel új kémiai terek irányába: szelektív és hatékony szintézisek
       Magyar Kémikusok Lapja 71, 185-185 (2016)
  16. Rita Megyesi, Enikő Forró, Ferenc Fülöp:
       Enzymatic Strategy for the resolution of new 1-hydroxymethyl tetrahydro-β-carboline derivatives in batch and continuous-flow systems
      ChemistryOpen 5, 254-260 (2016)
  17. Enikő Forró, Ferenc Fülöp:
       Cispentacin – Enzymatic highlights of its 25-year history
       Mini-Reviews in Organic Chemistry 13, 219-226 (2016)
  18. Zsófia Majláth, József Toldi, Ferenc Fülöp, László Vécsei:
       Excitotoxic mechanism in non-motor dysfunctions and levodopa-induced dyskinesia in Parkinson’s disease: the role of the interaction between
       the 
dopaminergic and the kynurenine system
       Current Medicinal Chemistry 23, 874-883 (2016)
  19. Nóra Török, Zsófia Majláth, Ferenc Fülöp, József Toldi, László Vécsei:
        Brain aging and disorders of the central nervous system: kynurenines and drug metabolism
       
Current Drug Metabolism17, 412-429 (2016)
  20. Ágnes Kasza, Ákos Hunya, Zsuzsa Frank, Ferenc Fülöp, Zsolt Török, Gábor Balogh, Miklós Sántha, Árpád Málind, Sándor Bernáth, Katie L.I.M.
        Blundell, Chrisostomos Prodromou, Ibolya Horváth, Hans-Joachim Zeiler, Philip L. Hooper, László Vigh, Botond Penke:
       Dihydropyridine derivatives modulate heat shock responses and have a neuroprotective effect in a transgenic mouse model of Alzheimer’s disease
       Journals of Alzheimer’s Disease53, 557-571 (2016)
  21. Beáta Fekete, Márta Palkó, István Mándity, Matti Haukka, Ferenc Fülöp:
        A domino ring-closure followed by retro-Diels-Alder reaction for the preparation of pyrimido[2,1-a]isoindole enantiomers
       Eur. J. Org. Chem. 3519-3527 (2016)
  22. Zsolt Galla, Enikő Forró, Ferenc Fülöp:
       Enhanced enzymatic synthesis of the enantiopure intermediate for the blockbuster drug intermediate abacavir through a two-step enzymatic
       cascade reaction
       Tetrahedron: Asymmetry 27, 729-731 (2016)
  23. M. Lukács, K. Warfvinge, L.S. Kruse, J. Tajti, F. Fülöp, J. Toldi, L. Vécsei, L. Edvinsson:
       KYNA analogue SZR72 modifies CFA-induced dural inflammation- regarding expression of pERK1/2 and IL-1β in the rat trigeminal ganglion
      The Journal of Headache and Pain 17:64, (2016)
  24. Judit Sas, István Szatmári, Ferenc Fülöp:
       One-pot α-arylation of β-carboline with indole and naphthol derivatives
      Current Organic Synthesis 13, 611-616 (2016)
  25. István Szatmári, Judit Sas, Ferenc Fülöp:
       C-3 functionalization of indole derivatives with isoquinolines
       Current Organic Chemistry 20, 2038-2054 (2016)
  26. Nóra Grecsó, Enikő Forró, Ferenc Fülöp, Antal Péter, István Ilisz, Wolfgang Lindner:
       Combinatorial effects of the configuration of the cationic and the anionic chiral subunits of four zwitterionic chiral stationary phases leading to
       reversal of elution order of cyclic β3-amino acid enantiomers as ampholytic model compounds
       Journal of Chromatography A 1467, 178-187 (2016)
  27. Gyula Lajkó, Nóra Grecsó, Rita Megyesi, Enikő Forró, Ferenc Fülöp, Denise Wolrab, Wolfgang Lindner, Antal Péter, István Ilisz:
        Enantioseparation of β-carboline derivatives on polysaccharide- and strong cation exchanger-based chiral stationary phases. A comparative study.
        Journal of Chromatography A 1467, 188-198 (2016)
  28. Gyula Lajkó, Timea Orosz, Loránd Kiss, Enikő Forró, Ferenc Fülöp, Antal Péter, István Ilisz:
        High-performance liquid chromatographic enantioseparation of fluorinated cyclic β3-amino acid derivatives on polisaccharide-based chiral
        stationary phases. Comparison with nonfluorinated counterparts
        Biomedical Chromatography30, 1441-1448 (2016)
  29. E. Marciniak, M. Hasiec, Ferenc Fülöp, T. Misztal:
       Salsolinol – a potential inhibitor of the gonadotropic axis in sheep during lactation
       Domestic Animal Endocrinology 58, 97-103 (2016)
  30. Renáta Anita Ábrahámi, Loránd Kiss, Pablo Barrio, Ferenc Fülöp:
        Synthesis of fluorinated piperidine and azepane β-amino acid derivatives
       Tetrahedron 72, 7526-7535 (2016)
  31. Amir Geramipour, Zsófia Kohajda, Claudia Corici, János Prorok, Zsolt Szakonyi, Kinga Oravecz, Zoltán Márton, Norbert Nagy, András Tóth, Károly
       Acsai, László Virág, András Varró, Norbert Jost:
       The investigation of the cellular electrophysiological and antiarrhytmic effects of a novel selective sodium–calcium exchanger inhibitor. GYKB
       6635, in canine and guinea-pig hearts
       Can. J. Physiol. Pharmacol94, 1090-1101 (2016)
  32. Enikő Forró, Rita Megyesi, Tihamér A. Paál, Ferenc Fülöp:
        Efficient dynamic kinetic resolution method for the synthesis of enantiopure 6-hydroxy- and 6-methoxy-1,2,3,4-terahydroisoquinoline-1
        carboxylic acid
        Tetrahedron: Assymetry 27, 1213-1216 (2016)
  33. Attila Márió Remete, Melinda Nonn, Santos Fustero, Ferenc Fülöp, Loránd Kiss:
        A stereocontrolled protocol to highly functionalized fluorinated scaffolds through a fluoride opening of oxiranes
       Molecules 21, 1493-1502
  34. Gyula Lajkó, Nóra Grecsó, Gábor Tóth, Ferenc Fülöp, Wolofgang Lindner, Antal Péter, István Ilisz:
       A comparative study of enantioseparations of Nα-Fmoc proteinogenic amino acids on Quinine-based zwitterionic and anion exchanger-type chiral
       stationary phases under hydro-organic liquid and subcritical fluid chromatographic conditions
       Molecules 21, 1579-1597 (2016)
  35. Antal Péter, Nóra Grecsó, Gábor Tóth, Ferenc Fülöp, Wolfgang Lindner István Ilisz:
        Ultra-trace analysis of enantiomeric impurities in proteinogenic N-Fmoc-acids samples on Cinchona alkaloid-based chiral stationary phases
        Israel Journal of Chemistry 56, 1042-1051 (2016)
  36. Yuki Inaba, Yuki Kato, Azumi Itou, Aoi Chiba, Ken Sawa, Ferenc Fülöp, György Miklós Nagy, Tsutomu Hashizume:
        Effects of extracerebral dopamine on salsolinol- or thyrotropin-releasing hormone-induced prolactin (PRL) secretion in goats
       Animal Science Journal 87, 1522-1527 (2016)
  37. Loránd Kiss, Melinda Nonn,Reijo Sillanpää, Matti Haukka, Santos Fustero, Ferenc Fülöp:
       Chemoselective, substrate-directed fluorination of functionalized cyclopentane β-amino acids
       Chemistry an Asian Journal 11, 3376-3381 (2016)
  38. Magyar Tímea, Ferenc Miklós, László Lázár, Ferenc Fülöp:
       Synthesis of 2-(hetero)arylquinazolinones in aqueous media
       Arkivoc VI, 247-258 (2016)